Galantide TFA
规格
Cas Number | G659296 |
规格或纯度 | ≥98% |
纯度 | ≥98% |
包装 | 1mg 或 5mg 或 500μg |
产品信息
品牌 | 阿拉丁 |
溶解性 | DMSO : 100 mg/mL (43.22 mM; Need ultrasonic) H2O : < 0.1 mg/mL (ultrasonic;adjust pH to 2 with HCl) (insoluble) |
过滤标签 | Neuropeptide Y Receptor,GPCR/G Protein,神经元信号传导 |
储存温度 | 避光,充氩,干燥,-80℃储存 |
运输条件 | 超低温冰袋运输 |
英文描述 |
Galantide TFA is a reversible and non-specific galanin (GAL) receptor antagonist. Galantide TFA dose-dependently shows antagonism to galanin-induced K + conductance with an IC 50 value of 4 nM. Galantide TFA can be used for the research of neurological di Appearance:Solid In Vitro:Galantide TFA (0.1-10000 nM) inhibits the galanin-induced activation of the K + conductance with an IC 50 value of 4 nM. Galantide TFA (0.1-10000 nM) dose-dependently inhibits the voltage-dependent Ba 2+ current with an IC 50 value of 16 nM. Gal In Vivo:Galantide TFA (5 nm; icv, once) inhibits luteinizing hormone (LH) release of ovariectomized (OVX) rats. Galantide TFA (1 and 5 nm; iv, for 3 times, at 1300, 1400 and 1500 h) decreases steroid-induced luteinizing hormone (LH) surge in estradiol benzoa Biological Activity:Galantide TFA is a reversible and non-specific galanin (GAL) receptor antagonist. Galantide TFA dose-dependently shows antagonism to galanin-induced K + conductance with an IC 50 value of 4 nM. Galantide TFA can be used for the research of neurological di |