Virodhamine
规格
| Cas Number | 287937-12-6 |
| 规格或纯度 | Moligand™, ≥98% |
| 级别 | Moligand™ |
| 纯度 | ≥98% |
| 包装 | 100mg 或 50mg 或 10mg 或 5mg 或 25mg |
产品信息
| 品牌 | 阿拉丁 |
| Action Type | 激动剂 |
| Mechanism Of Action | GPR55 激动剂 |
| 溶解性 | Soluble in Ethanol (supplied pre-dissolved in anhydrous ethanol, 5mg/ml) |
| 简短描述 | 内源性大麻素受体混合拮抗剂/激动剂 |
| 英文简短描述 | an endogenous cannabinoid receptor mixed antagonist/agonist |
| 过滤标签 | GPR55 Agonist,Cannabinoid Receptor,GPCR/G Protein,神经元信号传导 |
| 储存温度 | -20°C储存 |
| 运输条件 | 超低温冰袋运输 |
| 描述 |
内源性大麻素受体混合拮抗剂/激动剂的周边浓度高于anandamide。GPR55和CB2的完全激动剂和CB1的部分拮抗剂/激动剂（GPR55，CB2和CB1受体的EC | 50 |值分别为12、381和2920 nM）。在体内诱导体温过低。 |
| 英文描述 |
Endogenous cannabinoid receptor mixed antagonist/agonist found in higher concentrations peripherally than anandamide. Full agonist at GPR55 and CB2 and partial antagonist/agonist at CB1 (EC|50|values are 12, 381 and 2920 nM at GPR55, CB2 and CB1 receptors respectively). Induces hypothermia in vivo. |