DGY-06-116
规格
Cas Number | 2556836-50-9(DMSO) |
规格或纯度 | 10mM in DMSO |
包装 | 1ml |
产品信息
品牌 | 阿拉丁 |
浓度 | 10mM in DMSO |
溶解性 | Solubility (25°C) In vitro DMSO: 100 mg/mL (167.47 mM); Water: Insoluble; Ethanol: Insoluble; |
简短描述 | Src抑制剂 |
英文简短描述 | Src Inhibitors |
过滤标签 | Compound libraries |
储存温度 | -80℃储存 |
运输条件 | 超低温冰袋运输 |
生化和生理学机理 | DGY-06-116 是一种不可逆的共价选择性 Src 抑制剂,IC50 为 2.6 nM。 |
英文描述 |
Information DGY-06-116 DGY-06-116 is an irreversible covalent and selective inhibitor of Src with IC50 of 2.6 nM. Targets Src (Cell-free assay) 2.6 nM In vitro DGY-06-116 inhibits Src enzymatic activity. DGY-06-116 binds covalently to Src in a manner similar to SM1-71, where the p-loop must kink to establish the covalent bond. |