EML4-ALK kinase inhibitor 1
规格
Cas Number | 1373409-08-5 |
规格或纯度 | ≥98% |
纯度 | ≥98% |
包装 | 100mg 或 50mg 或 10mg 或 5mg 或 25mg |
产品信息
品牌 | 阿拉丁 |
溶解性 | DMSO : 110 mg/mL (189.41 mM; Need ultrasonic) |
过滤标签 | Anaplastic lymphoma kinase (ALK),Protein Tyrosine Kinase/RTK |
储存温度 | 避光,-20°C储存,干燥 |
运输条件 | 超低温冰袋运输 |
生化和生理学机理 | EML4-ALK 激酶抑制剂 1 是棘皮动物微管相关蛋白样 4-无性淋巴瘤激酶(EML4-ALK)的一种强效口服活性抑制剂,其 IC 50 为 1 nM。 |
英文描述 |
EML4-ALK kinase inhibitor 1 is a potent orally active inhibitor of echinoderm microtubule-associated protein-like 4-anaplastic lymphoma kinase (EML4-ALK) , with an IC 50 of 1 nM Form:Solid IC50& Target:IC50: 1 nM (EML4-ALK) |