Glucocorticoid receptor agonist-1
规格
Cas Number | 2166375-82-0 |
规格或纯度 |
包装 | 10mg 或 5mg |
产品信息
品牌 | 阿拉丁 |
过滤标签 | Glucocorticoid Receptor,Immunology/Inflammation,Vitamin D Related/Nuclear Receptor |
储存温度 | 2-8°C储存,避光 |
运输条件 | 冰袋运输 |
生化和生理学机理 | 糖皮质激素受体激动剂-1 是一种强效糖皮质激素受体激动剂,其 IC 50 为 2.8 nM,提取自专利 WO2017210471A1,即化合物 41。 |
英文描述 |
Glucocorticoid receptor agonist-1 is a potent glucocorticoid receptor agonist with an IC 50 of 2.8 nM extracted from patent WO2017210471A1, compound 41 In Vitro Glucocorticoid receptor agonist immunoconjugates are useful for treating autoimmune diseases such as, but not limited to, rheumatoid arthritis, juvenile idiopathic arthritis, psoriatic arthritis, ankylosing spondylitis, adult Crohn's disease, pediatric Crohn's disease, ulcerative colitis, plaque psoriasis, hidradenitis suppurativa, uveitis, Behcets disease, a spondyloarthropathy, or psoriasis. MCE has not independently confirmed the accuracy of these methods. They are for reference only. Form:Solid IC50& Target:IC50: 2.8 nM (Glucocorticoid receptor) |