马来酸甲硫基西平
规格
Cas Number | 19728-88-2 |
规格或纯度 | ≥98% |
纯度 | ≥98% |
包装 | 50mg |
产品信息
品牌 | 阿拉丁 |
溶解性 | Soluble in watere (5 mM). |
简短描述 | 有效的5-HT2和活性5-HT1拮抗剂 |
英文简短描述 | a potent 5-HT2 and active 5-HT1 antagonist |
过滤标签 | 5-HT Receptor,GPCR/G Protein,神经元信号传导 |
储存温度 | 室温 |
运输条件 | 常规运输 |
描述 |
马来酸噻吩并噻吩对5-HT | 5 |显示中等亲和力,对5-HT | 6 |和5-HT | 7 |显示高亲和力。马来酸噻吩并噻吩在5-HT | 1 |和5-HT | 2 |处也拮抗。有力的5-HT | 2 |拮抗剂,也具有5-HT | 1 |拮抗剂的活性。区分5-HT | 1D |子类型。 |
英文描述 |
Methiothepin maleate shows moderate affinity for 5-HT|5|and high affinity for 5-HT|6|and 5-HT|7|. Methiothepin maleate also antagonist at 5-HT|1|and 5-HT|2|. Potent 5-HT|2|antagonist, also active as 5-HT|1|antagonist. Differentiates 5-HT|1D|sub-types. |