Morphiceptin
规格
| Cas Number | 74135-04-9 |
| 规格或纯度 | ≥99% |
| 纯度 | ≥99% |
| 包装 | 10mg 或 1mg 或 5mg |
产品信息
| 品牌 | 阿拉丁 |
| 溶解性 | H2O : ≥ 250 mg/mL (479.29 mM) DMSO : 125 mg/mL (239.64 mM; Need ultrasonic) |
| 过滤标签 | Opioid Receptor,GPCR/G Protein,神经元信号传导 |
| 储存温度 | 干燥,-80℃储存 |
| 运输条件 | 超低温冰袋运输 |
| 生化和生理学机理 | Morphiceptin 是吗啡（μ）受体的强效特异性激动剂。Morphiceptin 作为一种合成肽，是牛奶蛋白 β-酪蛋白片段的酰胺。吗啡肽具有吗啡样活性，对吗啡（μ）受体具有高度特异性。 |
| 英文描述 |
Morphiceptin is a potent and specific agonist for morphine (μ) receptors . Morphiceptin, as a synthetic peptide, is the amide of a fragment of the milk protein β-casein. Morphiceptin has morphinelike activities and is highly specific for morphine (μ) receptors but not for enkephalin (⸹) receptors In Vivo Morphiceptin potently inhibits the binding of [ 3 H]dihydromorphine, 125 I-labeled FK33824, and [ 3 H]naloxone to rat brain membrane preparations with a 50 percent inhibition concentration (IC 50 ) of about 20 nM . MCE has not independently confirmed the accuracy of these methods. They are for reference only. Form:Solid IC50& Target:μ Opioid Receptor/MOR |