Pipequaline
规格
Cas Number | 77472-98-1(DMSO) |
规格或纯度 | 10mM in DMSO |
包装 | 1ml |
产品信息
品牌 | 阿拉丁 |
浓度 | 10mM in DMSO |
过滤标签 | GABA Receptor,神经元信号传导,膜转运器/离子通道,Compound libraries |
储存温度 | -80℃储存 |
运输条件 | 超低温冰袋运输 |
生化和生理学机理 | Pipequaline (PK 8165)是一种部分苯二氮卓受体激动剂,具有抗焦虑活性。 |
英文描述 |
Pipequaline (PK 8165) is a partial benzodiazepine receptor agonist with anxiolytic activity In Vivo Intravenously administered pipequaline exerts a partial suppression of activations by kainate, glutamate and acetylcholine. Microiontophoretic applications of pipequaline reduces the neuronal activation by kainate. Pipequaline produces dose-related decreases in motor activity. Pipequaline produces significant dose-related decreases in the number of head-dips made. MCE has not independently confirmed the accuracy of these methods. They are for reference only. IC50& Target:Benzodiazepine receptor |